2-Methylpropionate is a vitamin-B derivative also called thiamine disulfide. It is used in medicine for treatment of asthenia (weakness, loss of appetite and inability to concentrate). It is used as supplement by bodybuilders and athletes because it is believed to increase physical resistance to fatigue, improve neuromuscular efficiency, learning and memory, and improve metabolic function of the cerebral cortex. Some users have also reported improved sleep patterns after use of 2-methylpropionate supplements. Research shows that it improves energy levels by increasing choline uptake by hippocampal neurons, thus resulting in an increase in synthesis and release of acetylcholine. Its effects on brain are because it increases neuronal membrane permeability.

Caffeine is a central nervous system stimulant that temporarily wards off drowsiness and boosts alertness and energy.

Guarana Extract is the extract of the guarana plant. It contains a significant amount of guaranine, a substance that is similar to caffeine found in coffee beans. It helps stimulate the adrenal glands and increase the production and release of hormones such as epinephrine, norepinephrine (adrenaline), and dopamine. This helps the metabolism of the body that enhances fat loss, and increases energy and endurance. It helps the body burn the fats to be used for energy. It aids in fighting stress, weakness and fatigue. As a stimulant, it also improves mental alertness, clarity, focus, concentration, and memory retention. Guarana also also improves the libido or sex drive in both men and women. Guarana also contains tannins that help prevent diarrhea and soothes the digestive system.

Thiamine is a water-soluble vitamin with no known toxic effects if taken with other members of the vitamin B complex. Thiamine is essential to a strong appetite and to enable the body to use sugars and other carbohydrates.

Yohimbine HCL is a tryptamine alkaloid obtained from a medicinal herb Pausinystalia yohimbe, also known as yohimbe or yohimbe bark. This supplement belongs to the group of stimulant drugs, which has aphrodisiac qualities. Yohimbine chloride—a standardized form of yohimbine—is also used to treat erectile dysfunction. It can also be used to treat sexual side effects caused by some antidepressants (SRRIs), female hyposexual disorder and is also a blood pressure boosting agent and treats orgasmic dysfunction in men. Used orally as a supplement causes significant fat loss in athletes. Yohimbine is an alkaloid obtained from the bark of Pausinystalia yohimbe Pierre where the active ingredient yohimbine HCL (indole alkaloid) is obtained from.